Cardiac & Antihypertensive

Brinzolamide + Brimonidine TartrateThird Party Manufacturing in India

Looking to get Brinzolamide + Brimonidine Tartrate manufactured under your brand? Our WHO-GMP certified partner facilities support PCD franchise partners and global export opportunities structured across 25+ countries.

WHO-GMP Certified
Export Ready
PCD Franchise Available
CAS Number
138890-62-7
Drug Class
Carbonic Anhydrase Inhibitor and Alpha-2 Adrenergic Agonist Combination
Molecular Formula
Combination product (C₁₂H₂₁N₃O₅S₂ / C₁₁H₁₀BrN₅·C₄H₆O₆)
Molecular Weight
Combination product
Grade Standards
IP, BP, USP
Therapeutic Category
Cardiac & Antihypertensive
MOQ
10,000 vials per batch
Dosage Forms
Eye Drops

Mechanism of Action

Brinzolamide + Brimonidine Tartrate works by combining two distinct pharmacological actions to lower intraocular pressure in open-angle glaucoma. Brinzolamide inhibits carbonic anhydrase II in the ciliary processes, reducing bicarbonate ion secretion and subsequent sodium and fluid transport, which decreases aqueous humor production. Brimonidine tartrate acts concurrently as an alpha-2 adrenergic agonist, suppressing aqueous humor synthesis via G-protein pathways and enhancing uveoscleral outflow. Unlike traditional dual beta-blocker therapies, it avoids systemic cardiovascular side effects. It is highly effective and well-tolerated.

Therapeutic Uses & Indications

Therapeutic Uses

  • Advanced Glaucoma Management: Prescribed for patients requiring multi-mechanism intraocular pressure reduction when monotherapy fails.
  • Ocular Hypertension: Indicated for lowering intraocular pressure to mitigate the risk of optic nerve field defects.

Dosage Forms We Manufacture

Eye Drops
1.0% w/v + 0.2% w/v · 10mg + 2mg

Frequently Asked Questions

What is the minimum order quantity for Brinzolamide + Brimonidine Tartrate?
Minimum order quantity for Brinzolamide + Brimonidine Tartrate is 10,000 vials per batch. Please contact us for bulk pricing and custom quantities.
What dosage forms of Brinzolamide + Brimonidine Tartrate can you manufacture?
We manufacture Brinzolamide + Brimonidine Tartrate as: Eye Drops (1.0% w/v + 0.2% w/v, 10mg + 2mg).
Are your manufacturing facilities WHO-GMP certified?
Yes. Celesta Healthcare works exclusively with WHO-GMP certified partner production facilities. All manufacturing batches are subject to strict quality control and documentation.
Can you manufacture Brinzolamide + Brimonidine Tartrate for export?
Yes. We provide export-ready Brinzolamide + Brimonidine Tartrate formulations structured across 25+ countries. We provide full export documentation including Certificate of Analysis (CoA), Certificate of Origin, and regulatory dossiers on request.
What grade standards do you follow for Brinzolamide + Brimonidine Tartrate?
We manufacture Brinzolamide + Brimonidine Tartrate to IP, BP, USP pharmacopoeial standards.
Third Party Manufacturing

Get Brinzolamide + Brimonidine Tartrate made under your brand

  • WHO-GMP certified facilities
  • Quote within 24 hours
  • MOQ from 10,000 vials per batch
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+91 9689237122 · replies within hours

Our Manufacturing Capabilities

  • WHO-GMP Certified Partner Plants
  • 25+ years of pharma industry experience
  • PCD Franchise with monopoly rights
  • Export support across 25+ countries
  • Small batch to commercial scale
  • Custom formulation development

Packaging Options

Sterile dropper bottles with controlled dispensing tips. Packaging customized to client brand guidelines.

Start Manufacturing Brinzolamide + Brimonidine Tartrate Today

Celesta Healthcare provides WHO-GMP certified third-party manufacturing for Brinzolamide + Brimonidine Tartrate across all dosage forms. PCD franchise and export orders welcome.

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